Attention: Only available as part IRB approved INVESTIGATIONAL RESEARCH Studies with an Independent Data Safety Monitoring Board, Proper Adverse Event Reporting SOPs and Regulatory Compliant Informed Patient Consent. Only available at properly trained and compliant for Good Clinical Practices Clinical Trial Locations with qualified personnel with sufficient required database management skills.
Overview
In partnership with NudaLabs, Lionheart Health offers physician-guided, AI-personalized peptide protocols exclusively through qualified international (OUS) clinics. These advanced stacks are designed to support weight loss, cellular regeneration, immune health, and aging research—pushing the frontier of functional medicine with structured, supervised care. Contact us to get connected to a certified clinician at an enrolled Lionheart OUS location.
Key Benefits
These investigational protocols deliver targeted therapeutic support:
- Personalized peptide stacks based on full diagnostic review
- Investigational GLP-1 microdosing for weight loss and longevity
- Clinically guided by certified functional medicine experts
- Custom protocols for tissue regeneration, energy, immunity, and aging
- Delivered under IRB-approved research protocols in select countries
Bioelectric-Enhanced Peptide & Klotho-Up™ Regenerative Systems
At Lionheart Longevity, peptides are only the beginning. We combine precision peptide therapies with advanced Klotho signaling and bioelectric enhancement to support a next-generation regenerative framework designed to optimize how the body responds, repairs, and adapts.
- Peptides signal
- Bioelectricity activates
- Klotho coordinates system-wide repair
InstaMed® Regenerative Peptide Strips
Needle-free peptide delivery through convenient, pre-dosed oral dissolving strips.
Lionheart Longevity is expanding its peptide offerings to include InstaMed® Regenerative Peptide Strips, an oral dissolving strip platform designed for buccal, mouth-to-body delivery. The strips are pre-dosed, require no water or injection, and are available in multiple peptide formulations.
Why InstaMed® Peptide Strips
- Needle-free, pre-dosed delivery
- No water required
- Convenient and travel-friendly
- Individually packaged strips
- Designed for buccal/oral mucosal delivery
- Multiple peptide formulations across wellness and longevity applications
Available InstaMed® Formulations
Rebuild — BPC-157
Strength — CJC-1295 / Ipamorelin
Beauty & Hair — GHK-Cu
Immune — Thymosin Alpha-1
Intimacy — PT-141+
Energy — NAD+
Vitality — Glutathione + NAC
Metabolic — Ultratrutide™
Performance — Boost (MOTS-c)
Rest — Sleep (DSIP / GABA / 5-HTP)
Rejuvenation — KLOW
Focus — Neuro (Semax / Selank)
Explore InstaMed® Peptide Strips
InstaMed® products and peptide formulations are subject to applicable regulatory requirements and are intended for use only as permitted by applicable law and the relevant research or clinical protocol. Product availability may vary.
🧬 The Klotho-Up™ Advantage
Klotho is a master longevity regulator associated with:
- Cellular repair and regeneration
- Brain function and neuroprotection
- Muscle strength and endurance
- Vascular and kidney health
- Inflammation and oxidative stress balance
Unlike single-pathway approaches, Klotho is designed to support multi-system coordination of regenerative signaling.
⚡ Bioelectric-Enhanced Peptide Technology (Patent Pending)
Lionheart Health is advancing bioelectric-enhanced peptide delivery systems designed to improve how the body absorbs, distributes, and responds to peptides.
Integrated platforms include:
- BodStim™ (full-body EMS system)
- OrthoStim™ (targeted tissue repair)
- BrainBand™ (neuro-focused stimulation)
🔋 How Bioelectric Stimulation May Enhance Peptide Therapy
Bioelectric signaling is foundational to cellular communication and repair. When paired with peptides, it may:
- Increase cellular uptake of peptides
- Enhance receptor sensitivity and signaling response
- Improve blood flow and microcirculation
- Activate dormant regenerative pathways
- Support stem cell homing and retention
- Increase mitochondrial energy production
- Improve tissue conductivity and coordination
- Potentially reduce required dosing through improved efficiency
➡️ Result: More targeted, efficient, and amplified regenerative outcomes
💪 BodStim™ FDA-Cleared EMS Suit
Full-Body Bioelectric Acceleration of Peptide Protocols
The BodStim™ system is an FDA-cleared electrical muscle stimulation (EMS) suit designed to activate large muscle groups and systemic physiology—making it a powerful companion to peptide therapy.
🔬 Why BodStim™ Matters in Peptide Protocols
Peptides rely on circulation, receptor activation, and tissue responsiveness.
BodStim™ enhances all three.
⚡ How BodStim™ is Intended to Support Peptide Effectiveness
- Full-body circulation boost
→ Improves delivery of peptides to muscle, fat, and connective tissues - Muscle activation without joint strain
→ Stimulates fast- and slow-twitch fibers, enhancing anabolic signaling - Enhanced receptor engagement
→ Active tissue is more responsive to peptide signaling (GH, IGF-1, repair peptides) - Glucose uptake & metabolic activation
→ Supports GLP-1 / metabolic peptide pathways - Lymphatic movement and detox support
→ Helps clear inflammatory byproducts, improving recovery environment - Mitochondrial stimulation
→ Increases energy demand and utilization, synergizing with NAD+ and MOTS-C - Improved body composition signaling
→ Enhances fat metabolism and lean mass preservation - Neuromuscular re-education
→ Supports recovery in injury and aging-related muscle decline
🧠 System-Level Effect
BodStim™ turns the body into an “active biological receiver” for peptides.
➡️ Instead of passive delivery → dynamic, amplified response
🦁 Lionheart Protocol Integration
BodStim™ is used:
- 2x per week (typical protocol)
- Combined with peptide timing for maximum synergy
- Integrated with Klotho-Up™ programs to enhance systemic regeneration
➡️ Result: Faster strength gains, improved metabolic response, and deeper regenerative signaling
🧬 Klotho Peptides & Pathway Support
Lionheart focuses on enhancing Klotho expression and signaling, not just isolated peptide effects.
🔹 Klotho Pathway Support
MOTS-C • Epitalon • NAD+ • Thymosin Alpha-1
🔹 Regenerative Amplifiers
BPC-157 • TB-500 • GHK-Cu • IGF-1 variants
🔹 Hormonal & Metabolic Alignment
Sermorelin • Ipamorelin • CJC-1295 • GLP therapies
🔴 Core Peptide Categories
Healing & Repair – BPC-157 • TB-500 • GHK-Cu • KPV
Energy & Mitochondria – MOTS-C • SS-31 • NAD+ • 5-Amino-1MQ
Growth Hormone – Sermorelin • Ipamorelin • CJC-1295 • GHRPs
Fat Loss – Semaglutide • Tirzepatide • Cagrilintide • Retatrutide
Hormonal – Kisspeptin • HCG • HMG • IGF-1
Sleep & Longevity – DSIP • Epitalon • Thymosin Alpha-1
Pain & Nerve – ARA-290
🚀 Future of Longevity at Lionheart (INVESTIGATIONAL)
🧬 Klotho Nanotechnology
- Klotho Nanoflowers™ – Sustained, targeted regenerative signaling
🧠 Implantable & Wearable Systems
- KlothoImplant™ – Continuous internal delivery
- KlothoPod I™ – Wearable daily optimization
- KlothoPod II™ – Smart adaptive delivery system
- KlothoPatch™ – Transdermal peptide + bioelectric system
➡️ Moving from periodic therapy → continuous regeneration
α-Klotho Monoclonal Antibody (a-Klotho MAB), 10 mcg/vial, 2 vials product = $631
🦁 The Lionheart System
We combine:
- Peptides
- Klotho-Up™ signaling
- Bioelectric systems (BodStim™, OrthoStim™, BrainBand™)
- Regenerative biologics
- AI-driven personalization
- 460+ biomarker tracking
➡️ Outcome: Multi-system human optimization
⚠️ Important Note
BodStim™ is FDA-cleared for muscle stimulation, conditioning, and rehabilitation support.
Peptide and Klotho-Up™ protocols are part of personalized wellness and investigational programs under the Lionheart Klotho-Up Study under IRB and DSMB supervision. Requires informed patient consent. INVESTIGATIONAL RESEARCH.
Results vary based on individual biology and adherence.
“Don’t just take peptides. Activate your biology to respond to them.”
Klotho-Up™ + Bioelectric Enhancement | Only at Lionheart
Targeted Peptide Applications by System
❤️ Sexual Health Optimization
Performance, libido, and vascular function
- Enhances blood flow and endothelial function
- Supports nitric oxide signaling for performance
- Improves libido and hormonal signaling balance
- Supports erectile function and sexual responsiveness
- Aids recovery of reproductive tissue health
- May improve testosterone signaling and vitality
- Often combined with bioelectric stimulation (ErectiStim™ / FemStim™) for enhanced response
🧠 Brain Health & Cognitive Performance
Clarity, memory, mood, and neuroprotection
- Supports neuroplasticity and brain cell repair
- Enhances memory formation and recall
- Improves focus, clarity, and mental energy
- Helps regulate mood and stress response
- Supports mitochondrial energy production in neurons
- May protect against neuroinflammation and degeneration
- Often paired with BrainBand™ bioelectric stimulation for amplified effects
🦵 Joint Health & Musculoskeletal Support
Pain reduction, mobility, and structural repair
- Reduces inflammation in joints and connective tissue
- Supports cartilage, tendon, and ligament repair
- Enhances mobility and range of motion
- Accelerates recovery from injury or overuse
- Promotes collagen synthesis and structural integrity
- Helps reduce chronic pain signaling
- Synergizes with OrthoStim™ bioelectric therapy for deeper repair
🌿 Gut Health & Digestive Function
Inflammation control, microbiome balance, and repair
- Supports intestinal lining repair (“gut barrier”)
- Reduces gut inflammation and irritation
- Helps regulate immune activity in the GI tract
- Supports microbiome balance and digestive efficiency
- May improve symptoms of bloating, discomfort, and sensitivity
- Enhances nutrient absorption and metabolic signaling
- Often integrated with personalized nutrition protocols
👁️ Vision Health Support
Retinal protection, circulation, and cellular health
- Supports retinal cell protection and function
- Enhances microcirculation to ocular tissues
- Reduces oxidative stress in the eye
- May support visual clarity and focus
- Promotes cellular repair in aging eye structures
- Potential support for macular and optic nerve health
- Future integration with EyeCell™ and bioelectric stimulation platforms
👂 Hearing Health Support
Auditory function, nerve health, and regeneration
- Supports auditory nerve health and signaling
- May help protect against inflammation-related hearing decline
- Enhances microvascular circulation to inner ear structures
- Supports cellular repair in cochlear tissues
- May improve resilience to noise-induced stress
- Potential support for tinnitus-related pathways
- Future integration with bioelectric auditory stimulation technologies
“Precision peptides. System-wide impact. Bioelectric amplification.”
How It Works
Each protocol is developed through a collaboration between NudaLabs and Lionheart’s clinical team using AI analysis of diagnostic results. A typical investigational stack may include peptides such as GHK-Cu (skin and tissue regeneration), Epitalon (telomere and circadian support), Thymalin (immune rejuvenation), MOTS-c (mitochondrial health and metabolism), and FOXO4-DRI (senescent cell clearance – high research risk).
Peptide Pen & Cartridge System
A pharmaceutical-grade multi-dispense pen designed for the clinic. Pre-compounded cartridges, calibrated dial, sealed sterile filling. Hand it to a nurse and the protocol delivers itself.
- Pre-compounded cartridges: Peptides arrive sealed inside the cartridge with saline / Class 3 Pure Water — up to one year of stability without any bench prep.
- Calibrated dial system: Five dial positions deliver 0.15 – 0.75 mL with repeatable precision. Any tech can dispense at the chair without unit conversions.
- Up to 20 Dispense per cartridge: Built for protocols. Sell a starter pen, restock cartridges — recurring revenue without the compounding burden.
- Cross-formulation compatibility: One pen body, every stack. Professional users keep the pen between protocols — recovery, longevity, aesthetic, cognitive.
Interested in expanding your clinic’s offerings? Partner with us
FDA / REGULATORY & MEDICAL DISCLAIMER
FOR RESEARCH USE ONLY IN IRB APPROVED STUDIES with proper patient consent and oversight
This content is provided for educational, scientific and informational purposes only and is not intended as medical advice or as a claim that any product, therapy, protocol or combination described herein has been approved or cleared by the U.S. Food and Drug Administration (“FDA”) for the uses discussed.
Certain products, devices or components referenced by Lionheart Health® may have received FDA clearance or other regulatory authorization for specific indications. Such authorization should not be interpreted as FDA approval or clearance of other uses, modified applications, combination protocols, bioelectric signaling programs, regenerative medicine applications, peptide protocols or investigational therapies described on this website.
Some technologies, therapeutic applications, peptides, biologics, cellular therapies, bioelectric signaling protocols and combination approaches discussed by Lionheart Health may be investigational, under development, used solely for research, or not FDA-approved or FDA-cleared for the particular application described. References to laboratory studies, animal studies, pilot studies, IRB-reviewed research, clinical investigations, published literature or preliminary clinical observations should not be interpreted as establishing safety or effectiveness or as representing FDA authorization.
Investigational products and protocols are to be studied or used only in accordance with applicable federal and state law and, where required, appropriate FDA, IRB, IDE, IND or other regulatory oversight. Nothing on this website is intended to promote or commercially offer an investigational medical product in violation of applicable law.
Results described from research or clinical studies represent findings from the particular study populations, protocols and endpoints evaluated. Individual results may vary, and preliminary findings may not be confirmed in larger, randomized or independently replicated studies.
Lionheart Health does not represent that its complete multi-modality longevity, regenerative medicine or health-optimization programs have been evaluated, cleared or approved by the FDA as a whole. References to FDA-cleared devices or components apply only to the specific products and indications covered by their respective regulatory authorizations.
Treatment decisions should be made by an appropriately licensed healthcare professional based upon an individual patient’s medical history, condition, risks and potential benefits. Nothing contained on this website should replace consultation with a qualified healthcare provider.
For dietary supplements where applicable: These statements have not been evaluated by the Food and Drug Administration. This product is not intended to diagnose, treat, cure, or prevent any disease.
© Lionheart Health, Inc. All rights reserved.
What to Expect
During Treatment
After an in-person or virtual consult, approved patients begin a physician-supervised peptide therapy cycle using curated stacks and biomarker-based tracking.
After Treatment
Effects vary by peptide stack and use case but may include improved energy, lean mass preservation, reduced inflammation, and cognitive or metabolic support.
Ideal For
Peptide therapy is suitable for patients outside the U.S. participating in investigational longevity protocols. All patients must be under the care of a certified clinician at an enrolled Lionheart OUS location (Mexico, Costa Rica, Honduras, Antigua, or Dubai). Caution: Investigational use only. Not yet proven to be safe or effective.
IMPORTANT INVESTIGATIONAL USE NOTICE
The therapies described on this page are investigational and are available only as part of an IRB-approved research study conducted at trained clinical research locations operating in accordance with applicable Good Clinical Practice (GCP) requirements.
Participation requires appropriate informed patient consent and study oversight, including an Independent Data and Safety Monitoring Board (DSMB) where specified by the approved research protocol.